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TESOFENSINE
  • TESOFENSINE
  • TESOFENSINE
TESOFENSINE
$ 1,700.00 $ 3,000.00
$ 1,700.00 MXN
$ 1,445.00 MXN

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Tesofensine (NS 2330) is a synthetic phenyltropane derivative functioning as a triple monoamine reuptake inhibitor (TRI). It potently blocks the reuptake of dopamine (DAT), norepinephrine (NET), and serotonin (SERT) transporters. In neuropharmacology, this compound is utilized to model the modulation of synaptic neurotransmitter concentrations and central nervous system signaling pathways. Supplied as a pre-measured encapsulated reagent strictly for laboratory research and non-clinical analysis. Strictly for laboratory research use only.

CAS Number: 195875-84-4
Format: Encapsulated Monoamine Transporter Inhibitor

Chemical Description

Tesofensine is a serotonin–noradrenaline–dopamine reuptake inhibitor (SNDRI) belonging to the phenyltropane class of compounds. Chemically, it acts by binding to the presynaptic monoamine transporters (DAT, SERT, and NET), thereby preventing the clearance of neurotransmitters from the synaptic cleft. This mechanism leads to increased extracellular concentrations of dopamine, norepinephrine, and serotonin. It is widely used in neuroscience research to investigate the kinetics of triple reuptake inhibition and its downstream effects on central autonomic signaling pathways.

Research Applications

This compound is strictly for laboratory research use in the study of:

  • Neurotransmitter Transporter Kinetics: Investigation of the binding affinity (Ki) and inhibition constants (IC50) for dopamine, serotonin, and norepinephrine transporters in vitro.
  • Synaptic Signaling Modulation: Research into the sustained activation of post-synaptic receptors due to elevated monoamine availability in neuronal models.
  • Central Metabolic Signaling: In vitro analysis of sympathetic nervous system markers and thermogenic gene expression markers regulated by noradrenergic pathways.

Technical Specifications

  • Molecular Formula: C17H23Cl2NO
  • Molecular Weight: 328.3 g/mol
  • Class: Phenyltropane Derivative
  • Format: Research Capsule (Pre-measured for laboratory precision)
  • Purity: >99% (Active Ingredient)

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Presentation & Handling

  • Form: Oral capsules.
  • Storage: Store in a cool, dry environment, away from heat, light, and moisture.


Disclaimer: For Research Purposes Only

This content is provided strictly for laboratory research purposes and does not constitute an endorsement or recommendation for any non-laboratory application. The information provided regarding specific peptides is for educational and informational purposes only and must not be construed as medical, clinical, or legal guidance, nor as an encouragement for use in humans or animals.


Peptides described here are solely for use in structured scientific study by qualified researchers. We advise consulting with laboratory safety officers or research experts prior to handling these materials. The expectation of responsible, ethical utilization of this information for legitimate investigative and scholarly objectives is paramount. This notice governs all content on this site.

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